A PHASE I/II DOSE-ESCALATION AND EXPANSION STUDY EVALUATING THE SAFETY, PHARMACOKINETICS, AND ACTIVITY OF GDC-7035 AS A SINGLE AGENT AND IN COMBINATION WITH OTHER ANTI-CANCER THERAPIES IN PATIENTS WITH ADVANCED SOLID TUMORS WITH A KRAS G12D MUTATION

ENROLLING
Protocol # :
25-206
Conditions
Solid Tumor
Phase
I/II
Disease Sites
Neuroendocrine/Carcinoid
Gastroesophageal Junction
Gallbladder/Biliary
Other specified personal risk factors, not elsewhere classified
Lip, Oral Cavity and Pharynx
Esophagus
Stomach
Small Intestine
Colon
Rectum
Anus
Liver
Pancreas
Larynx
Lung
Other Respiratory and Intrathoracic Organs
Bones and Joints
Soft Tissue
Other Skin
Breast
Cervix
Corpus Uteri
Ovary
Other Female Genital
Prostate
Other Male Genital
Urinary Bladder
Kidney
Other Urinary
Eye and Orbit
Brain and Nervous System
Thyroid
Unknown Sites
Ill-Defined Sites
Other Endocrine System
Non-Hodgkin Lymphoma
Kaposi's Sarcoma
Melanoma, Skin
Principal Investigator
Park, Haeseong
Site Research Nurses
Arthur, Cara
Biddle, Elizabeth
Blake, Alyssa
Capulong, Florylene
Combs, Sarah
Grimes, Hayley
Speth, Celia
Treveloni, Emily
Vanasse, Richard

Trial Description

This is a first-in-human Phase I/II, open-label, multicenter, dose-escalation and
expansion study designed to evaluate the safety, pharmacokinetics, and preliminary
activity of GDC-7035 as a single agent and in combination with other anti-cancer
therapies in participants with advanced or metastatic solid tumors that harbor the KRAS
G12D mutation.

Eligibility Requirements

Inclusion Criteria:

- Histologically documented advanced or metastatic solid tumor with KRAS G12D mutation

- Agreement to adhere to the contraception requirements described in the protocol for
participants of childbearing potential and participants who produce sperm

Exclusion criteria:

- Malabsorption or other condition that would interfere with enteral absorption

- Active brain metastases

- Clinically significant cardiovascular dysfunction or liver disease

25-206